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CF53, MedChemExpress
MedChemExpress CF53 is a highly potent, selective and orally active inhibitor of BET protein, with a Ki of Kd of 2.2 nM and an IC50 of 2 nM for BRD4 BD1. CF53 binds to both the BD1 and BD2 domains of BRD2, BRD3, BRD4, and BRDT BET proteins with high affinities, very selective over non-BET bromodomain-containing proteins. CF53 shows potent anti-tumor activity both in vitro and in vivo.
515.70 EUR - 2301.75 EUR
Specifications
| Chemical Name or Material | CF53 |
|---|---|
| CAS | 1808160-52-2 |
| Color | Light Yellow |
| Purity Grade Notes | Research |
| Molecular Formula | C24H25N7O2 |
| Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
|---|---|---|---|---|---|---|---|---|---|
| Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
|
16470947
|
Medchem Express
HY-112610 |
50 mg |
1701.00 EUR
50mg |
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|
16464658
|
Medchem Express
HY-112610 |
10 mg |
773.55 EUR
10mg |
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|
16437377
|
Medchem Express
HY-112610 |
5 mg |
515.70 EUR
5mg |
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|
16435496
|
Medchem Express
HY-112610 |
100 mg |
2301.75 EUR
100mg |
Please sign in to purchase this item. Need a web account? Register with us today! | |||||
Description
CF53 is a highly potent, selective and orally active inhibitor of BET protein, with a Ki of Kd of 2.2 nM and an IC50 of 2 nM for BRD4 BD1. CF53 binds to both the BD1 and BD2 domains of BRD2, BRD3, BRD4, and BRDT BET proteins with high affinities, very selective over non-BET bromodomain-containing proteins. CF53 shows potent anti-tumor activity both in vitro and in vivo.Specifications
| CF53 | |
| Light Yellow | |
| C24H25N7O2 | |
| COC1=C(C2=C(C)ON=C2C)C=C(NC3=C4C(NC5=CC(C6CC6)=NN5C)=NC(C)=N3)C4=C1 | |
| 443.5 | |
| Research | |
| Cancer-programmed cell death |
| 1808160-52-2 | |
| Research | |
| DMSO : 110 mg/mL (248.03 mM; Need ultrasonic) | |
| 443.5 | |
| 98.09% | |
| Solid |
Safety and Handling
missing translation for 'shelfLife' : -20°C, stored under nitrogen∣In solvent : -80°C, 6 months∣-20°C, 1 month (stored under nitrogen)
Recommended Storage : -20°C, stored under nitrogen∣In solvent : -80°C, 6 months∣-20°C, 1 month (stored under nitrogen)
Research purposes only
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Product Title
CF53, MedChemExpress